Galeterone (TOK-001), TOK-001 help

BitterDB id=1720
Detailed experimental validation described in the associated resource.

References for the compound bitterness help

Resource Comment
[1] Fierro F. et al. Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands, Cellular and Molecular Life Sciences, 2023, 80, 114 PubMed 37012410

Known bitter receptors targets: help

Receptor Name Effective concentration (μM) EC50 (μM) References
Human  hTas2r14 3.0 PubMed:37012410

Sensory data about the compound bitterness: help

There is no sensory data available

Properties: help

388.5451 [g/mol] 4.85220
1 2
2 6
1

Identifiers: help

C26H32N2O
PAFKTGFSEFKSQG-PAASFTFBSA-N

Links:

[1] 11188409
[2] ZINC000006718442