LDE225 Diphosphate help

BitterDB id=1711
Detailed experimental validation described in the associated resource.

References for the compound bitterness help

Resource Comment
[1] Fierro F. et al. Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands, Cellular and Molecular Life Sciences, 2023, 80, 114 PubMed 37012410

Known bitter receptors targets: help

Receptor Name Effective concentration (μM) EC50 (μM) References
Human  hTas2r14 3.0 PubMed:37012410

Sensory data about the compound bitterness: help

There is no sensory data available

Properties: help

681.4885 [g/mol] 5.64570
1 10
3 4
7

Identifiers: help

C26H32F3N3O11P2
RWIVSVMMGFFZIJ-VWDRLOGHSA-N

Links:

[1] 45138699