Orantinib (TSU-68, SU6668), TSU-68 (SU6668,Orantinib) help

BitterDB id=1695
Detailed experimental validation described in the associated resource.

References for the compound bitterness help

Resource Comment
[1] Fierro F. et al. Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands, Cellular and Molecular Life Sciences, 2023, 80, 114 PubMed 37012410

Known bitter receptors targets: help

Receptor Name Effective concentration (μM) EC50 (μM) References
Human  hTas2r14 1.0 PubMed:37012410

Sensory data about the compound bitterness: help

There is no sensory data available

Properties: help

310.3471 [g/mol] 2.48530
2 1
2 3
4

Identifiers: help

C18H18N2O3
NHFDRBXTEDBWCZ-ZROIWOOFSA-N

Links:

[1] 5329099
[2] ZINC000003834032